An Orthogonal C-H Borylation – Cross-Coupling Strategy for the Preparation of Tetrasubstituted “A2B2”-Chrysene Derivatives with Tuneable Photophysical Properties

Kane W J Heard,  John J Morrison,  Laura Weston,  Chi H Lo,  Lucian Pirvu,  James Raftery,  Mark S Little,  Joseph J W McDouall,  Peter Quayle,  Stephen G Yeates
University of Manchester


Abstract

Phenacenes (cata-fused acene analogues) are of emerging interest in organic electronics, demonstrating potential as semiconducting materials and OLED emissive layers whilst maintaining oxidative stability.(1) In this study we introduce a cross coupling strategy for the orthogonal, A2B2, tetrasubstitution of chrysene allowing effective tuning of its photophysical properties.

Though our recently developed BHQ reaction we were readily able to access 4,10-dichlorochrysene.(2) Iridium catalysed C-H borylation(3) of 4,10-dichlorochrysene resulted in diborylation, affording as a single regioisomer the 2,8-diboryl-4,10-dichlorochrysene. The chlorine acts as removable steric directing group(4, 5) enabling ready access to 2,8- and 4,10- A2B2- tetrasubstituted chrysene derivatives.

After the initial C-H borylation, substitution of the 2,8- positions could then be performed with preservation of the 4,10-dichloro functionality, installing 4-(n-hexyl)phenyl, 4-(n-hexyloxy)phenyl, 4-(diphenylamino)phenyl and trifluoromethyl substituents. The remaining 4,10-dichloro positions were then accessed in subsequent palladium catalysed Kumada couplings in three examples, firstly installing phenyl and 2-thienyl substituents in the 4-(n-hexyl)phenyl substituted chrysene and then functionalising the 2,8-trifluoromethlated chrysene with 4-(diphenylamino)phenyl substituents to generate an orthogonally substituted donor-acceptor chrysene. This was of particular note as it was computationally predicted (TD-DFT) to possess a charge-transfer(6) transition from the HOMO to the LUMO due to its donor-acceptor structure.

The chrysene derivatives synthesised featured broadened UV-vis spectra particularly in the 2,8-Bis(4-(diphenylamino)phenyl) chrysene and the donor-acceptor substituted chrysene. Estimations of the HOMO and LUMO levels based on UV-vis optical band gap and CV data indicated increased HOMO levels and decreased band gaps, comparable with other contemporary p-type materials such as Pentacene, DNTT and Rubrene.(7) This is particularly notable in the case of the donor-acceptor chrysene and in the more electron rich derivatives featuring 2-thienyl and 4-(diphenylamino)phenyl functionalities.

In conclusion we present a novel and versatile strategy for the orthogonal synthesis of A2B2- tetrasubstituted chrysenes utilising a regioselective C-H borylation, resulting in a variety of derivatives with properties comparable to literature benchmarks, with possible applications either as p-type semiconductors or as tuneable emissive materials in OLEDs.

References:

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